Stephania Extract Cepharanthine Powder

Igoa Oloa: Stephania Japonica Extract
Fa'aLatina: Stephania cephalantha Hayata(Stephania japonica (Thunb.)Miers)/ Stephania epigaea Lo/ Stephania yunnanensis HSLo.
Fa'aaliga: Pa'epa'e, Efuefu Pa'epa'e Pa'u
Mea gaogao: Cepharanthine 80% -99% HPLC
Vaega Fa'aaogaina: Tuber/Root
Fa'aoga: oloa tau soifua maloloina
Liu liusuavai:145-155°
Ta'amilosaga fa'apitoa: D20+277°(c=2inchloroform)
Mea fa'apuna: 654.03°C (fa'atatau fa'atatau)
Malosi:1.1761(fa'atatau)
Fa'ailoga fa'atusa:1.5300(fa'atatau)
Tulaga teuina: underinertgas (nitrogen poʻo Argon) ile2-8°C
Solubility: Solu i le SO(35mg/mL) po'o le ethanol(20mg/mL)
Fa'asa'o (pKa):7.61±0.20(Va'ai)


Fa'amatalaga Oloa

Isi Fa'amatalaga

Faailoga o oloa

Folasaga o oloa

Stephania Extract Cepharanthine Powder o se mea e maua mai i fatu o le laau Stephania cephalantha Hayata(Stephania japonica (Thunb.) Miers) poʻo Stephania epigaea Lo/ Stephania yunnanensis HSLo.O le Cepharanthine ose oloa fa'anatura e tu'ufua mai lenei la'au ma ua avea ma autu o su'esu'ega 'ese'ese ona o ana mea tau vaila'au.Ua maua e fa'aalia ai gaioiga anti-SARS-CoV-2, fa'aalia le aoga i le taofiofia o le fa'ateleina o viral.E le gata i lea, ua faʻaalia e le Cepharanthine le malosi e toe faʻafoʻi ai le P-glycoprotein (P-gp)-mediated multidrug resistance i nisi sela ma faʻaleleia le lagona o vailaʻau faʻamaʻi i faʻataʻitaʻiga faʻataʻitaʻiga.E le gata i lea, ua faʻaalia e iai aʻafiaga faʻalavelave i le ate o le tagata cytochrome P450 enzymes CYP3A4, CYP2E1, ma le CYP2C9, ma e fesoʻotaʻi ma aʻafiaga antitumor, anti-inflammatory, ma antinociceptive.
I le aotelega, Stephania Extract Cepharanthine Powder o se paʻu paʻu o le oloa faʻanatura Cepharanthine e maua mai i le Stephania cephalantha laau, lea na faʻaalia ai le gafatia i le tele o faʻaoga faʻafomaʻi.

Fa'amatalaga(COA)

Oloa Cepharanthine
CAS 481-49-2
Su'ega 80%~99%
Fa'aaliga Pa'epa'e pa'epa'e
afifiina 1KG/Foil taga
Aitema Fa'amatalaga
Fa'aaliga efuefu pa'epa'e pa'epa'e, le manogi manogi, maualuga hygroscopic
Fa'ailoaga TLC: Fofo masani ma vaifofo su'ega nofoaga tutusa, RF
Su'esu'ega (Fa'amamago) 98.0%--102.0%
Fa'apitoa Optical -2.4°~ -2.8°
PH 4.5~7.0
Metala Mamafa (E pei o le Pb) ≤10ppm
As ≤1ppm
Pb ≤0.5ppm
Cd ≤1ppm
Hg ≤0.1ppm
Mea fa'atatau Ole nofoaga e le sili atu nai lo le tulaga masani ole fofo
Soli totoe <0.5%
Suavai Suavai <2%

Oloa Fa'ailoga

Stephania Extract Cepharanthine Powder o se oloa faʻanatura e maua mai le laau Stephania cephalantha Hayata.Ua maua le tele o mea tau vailaau, e aofia ai:
1. Gaoioiga Anti-SARS-CoV-2
2. Aafiaga faʻalavelave i le faʻateleina o viral
3. Fa'aliliuina ole P-glycoprotein-mediated multidrug resistance
4. Faʻaleleia atili o le faʻalogo i vailaʻau faʻamaʻi
5. Aafiaga fa'alavelave ile ate o le tagata cytochrome P450 enzymes CYP3A4, CYP2E1, ma le CYP2C9
6. Antitumor, anti-inflammatory, ma aʻafiaga antinociceptive

O le a le Biosynthesis o le Cepharanthine?

O le biosynthesis o le cepharanthine i Stephania e amata i le condensation o le dopamine ma le 4-hydroxyphenylacetaldehyde (4-HPAA, 5) e ala i le norcoclaurine synthase (NCS), e maua ai le norcoclaurine.

O le a le solubility o le Cepharanthine?

O le Cepharanthine e mafai ona solu i so'o so'o e pei ole ethanol, DMSO, ma le dimethyl formamide (DMF).O le solubility o le cepharanthine i nei solvents e tusa ma le 2, 5, ma le 10 mg / ml, i le faasologa.O le Cepharanthine e itiiti lava le solu i totonu o le vai.

Talosaga

O pisinisi talosaga mo Stephania Extract Cepharanthine Powder e aofia ai Pharmaceutical, Nutraceutical, Biotechnology, ma Herbal Medicine, o talosaga autu e pei ona taua i lalo:
Fa'aaogaina fa'apitoa i togafitiga fa'ama'i
Avanoa e fai ma fesoasoani i togafitiga o le kanesa
Avanoa mo le faʻaaogaina i togafitiga faʻamaʻi
Avanoa e avea o se vailaʻau faʻamaʻi
O nei talosaga e faʻamaonia ai le tele o faʻaogaina o le Stephania Extract Cepharanthine Powder i faʻalapotopotoga faʻapitoa.


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    2. Aveesea
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